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TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3550 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3550 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
HIV Protease
AChR
Dopamine Receptor
COX
Histamine Receptor
VEGFR
Sodium Channel
Parasite
Potassium Channel
EGFR
Calcium Channel
PI3K
PDE
Antifungal
Topoisomerase
HCV Protease
CDK
FLT
Cytochromes P450
PDGFR
Dehydrogenase
JAK
SARS-CoV
FGFR
PPAR
Microtubule Associated
c-Kit
Glucocorticoid Receptor
Reactive Oxygen Species
Ferroptosis
HDAC
mTOR
c-Met/HGFR
Influenza Virus
GABA Receptor
Src
Estrogen/progestogen Receptor
HBV
NF-κB
Mitophagy
Reverse Transcriptase
Prostaglandin Receptor
RAAS
Tyrosine Kinases
Nucleoside Antimetabolite/Analog
Adenosine Receptor
GPCR
Androgen Receptor
Raf
Proteasome
iGluR
Bcr-Abl
NMDAR
Serotonin Transporter
Epigenetic Reader Domain
GluR
Phosphatase
Virus Protease
PARP
TRP/TRPV Channel
ROS
HSV
Akt
Transferase
Aurora Kinase
Beta Amyloid
p38 MAPK
Estrogen Receptor/ERR
Norepinephrine
HSP
Progesterone Receptor
IL Receptor
ALK
MEK
HIF/HIF Prolyl-Hydroxylase
ATPase
Antiviral
c-RET
TNF
Histone Methyltransferase
Antioxidant
Opioid Receptor
DPP-4
Cholinesterase (ChE)
P-gp
Trk receptor
HER
Carbonic Anhydrase
Antifection
TLR
ribosome
GSK-3
PKC
ERK
CXCR
Endothelin Receptor
MMP
c-Fms
DNA Alkylator/Crosslinker
MAO
CCR
Chk
Interleukin
Retinoid Receptor
TAM Receptor
S1P Receptor
E1/E2/E3 Enzyme
Gamma-secretase
Mitochondrial Metabolism
Bcl-2 Family
AMPK
Syk
Thrombin
p53
Thyroid hormone receptor(THR)
Proton pump
DNA-PK
LPL Receptor
Wnt/beta-catenin
Caspase
SGLT
STAT
Phospholipase
HIF
CFTR
Integrin
Antifolate
Guanylate cyclase
Nrf2
Neurokinin receptor
FAK
NO Synthase
NADPH
CSF-1R
P2X Receptor
Hedgehog/Smoothened
DNA Alkylation
Lipoxygenase
IGF-1R
PLK
BTK
DHFR
P2Y Receptor
Reductase
Glutathione Peroxidase
MRP
ROCK
IAP
Vasopressin Receptor
OX Receptor
TGF-beta/Smad
RSV
ATM/ATR
Hydroxylase
Cannabinoid Receptor
HMG-CoA Reductase
S6 Kinase
ROS Kinase
Mdm2
PKA
GNRH Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Monoamine Oxidase
ADC Cytotoxin
Histone Demethylase
Factor Xa
Pim
Serine Protease
FXR
Aryl Hydrocarbon Receptor
RIP kinase
Drug Metabolite
Glucosidase
Smo
Xanthine Oxidase
DNA
Beta-Secretase
Aminopeptidase
Sirtuin
Casein Kinase
Ligand for E3 Ligase
DNA Methyltransferase
Sigma receptor
Kinesin
NOS
ROR
Amino Acids and Derivatives
BACE
JNK
Glucokinase
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
IRAK
AhR
CETP
Leukotriene Receptor
IDO
Glucagon Receptor
MT Receptor
Molecular Glues
Fatty Acid Synthase
Acyltransferase
Ephrin Receptor
CRFR
GHSR
Complement System
Gap Junction Protein
Ras
Chloride channel
PROTACs
MTP
CRM1
DprE1
YAP
LTR
IFNAR
Tie-2
Melatonin Receptor
Cholecystokinin Receptor
Photosensitizer
Liver X Receptor
Cysteine Protease
DNA gyrase
GlyT
Monoamine Transporter
IKZF
Neuropeptide Y Receptor
FAAH
CaMK
Wee1
PGE Synthase
MAPK
OAT
Decarboxylase
Neprilysin
Acetyl-CoA Carboxylase
Melanocortin Receptor
CGRP Receptor
NADPH-oxidase
Kras
NEDD8
Arginase
Cell wall
PERK
CaSR
Rho
PYK2
NAMPT
Glutaminase
Myosin
Annexin A
UGT
ABC Transporter
Somatostatin
KSP
DUB
Telomerase
STING
Free radical scavengers
GPCR19
LPA Receptor
PDK
Adenosine Deaminase
NOD
Tyrosinase
Protease-activated Receptor
NOD-like Receptor (NLR)
Imidazoline Receptor
PD-1/PD-L1
Taste receptor
GSNOR
Ligands for Target Protein for PROTAC
DYRK
VDA
Galectin
c-Myc
Serine/threonin kinase
IRE1
LDL
Na-K-Cl cotransporter
Hexokinase
Integrase
HCN Channel
Stearoyl-CoA Desaturase (SCD)
Epoxide Hydrolase
ATP Citrate Lyase
BCRP
Porcupine
CD73
transporter
PAI-1
GST
Oxytocin Receptor
Discoidin Domain Receptor (DDR)
p97
MLK
Apelin receptor
Advanced Glycation End Products
MicroRNA
Adenylyl Cyclase
Monocarboxylate transporter
NPC1L1
Hydrogenase
MALT
ASBT
Factor VIIa
Arrestin
Lipase
MIF
TOPK
GTPase
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
Neurotensin Receptor
Stemness kinase
SIK
FLAP
PAFR
Fas/FasL
GRK
Phosphorylase
Anion Exchanger
PROTAC Linker
Thioredoxin
ACK1
Cadherin
Lipid
Huntingtin
PSMA
Survivin
MNK
Histone Acetyltransferase
GluCls
ASK
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
Aromatase
PI4K
KLF
CRISPR/Cas9
Aquaporin
RXFP receptor
SGK
Anti-infection
BMI-1
PKM
Vitamin
Drug-Linker Conjugates for ADC
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