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IGF-1R
Cat.No. Product Name Information Area
T6943 Picropodophyllin (PPP) Picropodophyllin (PPP) is a selective IGF-1R inhibitor with IC50 of 1 nM. Phase 1/2. Others
T2693 AG1024 AG-1024 (Tyrphostin) inhibits IGF-1R autophosphorylation with IC50 of 7 μM, less pote... Other
T6419 BMS-536924 BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modes... Cancer
T6080 NVP-AEW541 NVP-AEW541 is a potent inhibitor of IGF-1R/InsR with IC50 of 150 nM/140 nM, greater p... Cancer
T2107 NVP-ADW742 NVP-ADW742 is an IGF-1R inhibitor with IC50 of 0.17 μM, >16-fold more potent again... Cancer
T6017 OSI-906 (Linsitinib) OSI-906 (Linsitinib) is a selective inhibitor of IGF-1R with IC50 of 35 nM; modestly ... Cancer
T6003 GSK1904529A GSK1904529A is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM, >... Cancer
T3079 GSK1838705A GSK1838705A is a potent IGF-1R inhibitor with IC50 of 2.0 nM, modestly potent to IR a... Cancer
T2491 AZ5104 AZ5104, the demethylated metabolite of AZD-9291, is a potent EGFR inhibitor with IC50... Cancer
T2349 BMS-754807 BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.... Cancer
T2085 PQ401 PQ401 inhibits autophosphorylation of IGF-1R domain with IC50 of <1 μM. Cancer
T1791 LDK378(Ceritinib) Ceritinib is an orally available inhibitor of the receptor tyrosine kinase activity o... Cancer
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