||Inhibitor of mitochondrial pyruvate dehydrogenase kinase (PDK). Shifts pyruvate metab...
||OSU-03012 (AR-12) is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM in a c...
||PHT-427 is a dual Akt and PDPK1 inhibitor (high affinity binding for the PH domains o...
||GSK2334470 is a novel PDK1 inhibitor with IC50 of ~10 nM in a cell-free assay, with n...
||BX-912 is a selective inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1) with ...
||BX795 is a potent and specific PDK1 inhibitor with IC50 of 6 nM, 140- and 1600-fold m...