info@targetmol.com    Tel: (857) 239-0968 / (617) 419-7131
Home > PI3K
PI3K
Cat.No. Product Name Information Area
T3986 SF2523 SF2523 is a highly selective and potent inhibitor of PI3K and BRD4with IC50 values of... Cancer
T3985 GDC-0326 GDC-0326 is a potent and selective inhibitor of α-Isoform of Phosphoinositide 3-Kinas... Others
T3705 GDC-0084 GDC-0084, also known as RG7666, is a phosphatidylinositol 3-kinase (PI3K) inhibitor w... Cancer
T3692 GNE 477 GNE-477 is a potent and efficacious dual PI3K/mTOR inhibitor with IC50 of 4 nM for PI... Others
T3348 PIK-293 PIK-293 is a PI3K inhibitor, mostly for PI3Kδ with IC50 of 0.24 μM, 500-, 100- and 50... Others
T3656 PKI-402 PKI-402 is a potent dual pan-PI3K/mTOR inhibitor targeting PI3Kα/β/γ/δ and mTOR with ... Others
T7015 VPS34-IN1 Vps34-IN1 is a potent and highly selective Vps34 inhibitor with IC50 of 25 nM invitro... Others
T7014 Voxtalisib (XL765, SAR245409) Voxtalisib (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ with... Others
T6945 PIK-III PIK-III, which is a selective inhibitor of ?VPS34 enzymatic activity, inhibits autoph... Others
T6938 PF-4989216 PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM,... Others
T6850 GSK2292767 GSK2292767 is a potent and selective PI3Kδ inhibitor. Others
T6845 GNE-317 GNE-317 is a potent, brain-penetrant PI3K inhibitor. Others
T6774 AZD8835 AZD8835 ia a novel mixed inhibitor of PI3Kα and PI3Kδ with IC50 of 6.2 nM and 5.7 nM,... Others
T6773 AZD8186 AZD8186 is a potent and selective inhibitor of PI3Kβ and PI3Kδ with IC50 of 4 nM and ... Others
T6757 AMG319 AMG319 is a potent and selective PI3Kδ inhibitor with IC50 of 18 nM, >47-fold selecti... Others
T3410 Momordin Icnew Momordin Ic might represent a potential anticancer activity, by inducing apoptosis th... Others
T1988 IPI-145 Duvelisib (IPI-145, INK1197) is a novel and selective PI3K δ/γ inhibitor with Ki and ... Cancer
T6704 TG100713 TG100713 is a pan-PI3K inhibitor against PI3Kγ, PI3Kδ, PI3Kα and PI3Kβ with IC50 of 5... Cancer
T6433 CAY10505 CAY10505 is dehydroxyl of AS-252424, which is a PI3Kγ inhibitor with IC50 of 33 nM. Cancer
T6394 AS-604850 AS-604850 is a selective, ATP-competitive PI3Kγ inhibitor with IC50 of 250 nM, over 8... Cancer
T6251 PF-04691502 PF-04691502 is an ATP-competitive PI3K(α/β/δ/γ)/mTOR dual inhibitor with Ki of 1.8 nM... Cancer
T6208 AS-252424 AS-252424 is a potent and selective inhibitor of PI3Kγ with IC50 of 33 nM; >10 fold s... Cancer
T6168 ZSTK474 ZSTK474 inhibits class I PI3K isoforms with IC50 of 37 nM, mostly PI3Kδ. Phase1/2. Immunology/ Cancer
T6143 PI-103 PI-103 is a multi-targeted PI3K inhibitor for p110α/β/δ/γ with IC50 of 2 nM/3 nM/3 nM... Cancer
T6110 YM201636 YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p110α an... Cancer
T6103 VS-5584 (SB2343) VS-5584 (SB2343) is a potent and selective dual PI3K/mTOR inhibitor for mTOR, PI3Kα/β... Cancer
T6087 AZD6482 AZD6482 is a PI3Kβ inhibitor with IC50 of 10 nM, 8-, 87- and 109-fold more selective ... Cancer
T6072 BGT226 (NVP-BGT226) BGT226 (NVP-BGT226) is a novel class I PI3K/mTOR inhibitor for PI3Kα/β/γ with IC50 of... Cancer
T2682 Acalisib (GS-9820) Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kδ with IC50 value of 12... Cancer
T2672 TG100-115 TG100-115 is a PI3Kγ/δ inhibitor with IC50 of 83 nM/235 nM, with little effect on PI3... Cancer
1