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Home > Tyrosine-Kinase-Adaptors-Others
Tyrosine-Kinase-Adaptors-Others
Cat.No. Product Name Information Area
T3962 TPI-1 TPI-1 is a SHP-1 inhibitor;? inhibits recombinant SHP-1 with an IC50 of 40 nM. Others
T3569 SU 5214 SU 5214 is a modulator of tyrosine kinase signal transduction. Others
T3710 XMD16-5 XMD16-5 is a tyrosine kinase nonreceptor 2(TNK2) inhibitor. TNK2 mutations have been ... Cancer
T3709 XMD8-87 XMD8-87 is a TNK2 inhibitor. XMD8-87 showed activity in the inhibition of TNK2 phosph... Cancer
T3160 HUHS015 HUHS015 is a potent PCA-1/ALKBH3 inhibitor. The bioavailability of HUHS015 was 7.2% i... Others
T3312 AM-2394 AM-2394 is a potent and selective Glucokinase agonist (GKA), which catalyzes the phos... Others
T3403 Glabridinnew Glabridin may serve as an anti-inflammatory agent in diabetes-related vascular dysfun... Others
T3337 Ddr1-In-1 DDR1-IN-1 is a potent and selective?discoidin domain receptor 1 (DDR1)?receptor tyros... Others
T3209 AMG-337 AMG-337 is a potent and highly selective small molecule ATP-competitive MET kinase in... Cancer
T2709 TAK901 TAK-901 is a novel inhibitor of Aurora A/B with IC50 of 21 nM/15 nM. It is not a pote... Cancer
T2659 GW2580 GW2580 is an orally bioavailable inhibitor of c-FMS kinase; completely inhibited huma... Cancer
T2457 IRAK-1-4 Inhibitor I IRAK-1-4 Inhibitor I is an inhibitor of both IRAK-1 and IRAK-4 with IC50 values of 0.... Cancer
T2328 Radotinib Radotinib, and sometimes referred to by its investigational name IY5511, is a drug fo... Cancer
T2281 GSK-2256098 A small molecule FAK kinase inhibitor, GSK2256098, inhibits growth and survival of pa... Cancer
T2153 1-NM-PP1 1NM-PP1(PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selec... Cancer
T2037 TH588 TH588 is first-in-class nudix hydrolase family inhibitor that potently and selectivel... Cancer
T2005 TP0903 TP-0903 is a potent and selective Axl kinase inhibitor with IC50 of 27 nM. Cancer
T1991 ZM323881 hydrochloride ZZZM 323881 hydrochloride is a potent and selective VEGFR2 inhibitor with IC50 of <2 ... Other
T1844 KPT-330 KPT-330 inhibited proliferation and induced cell cycle arrest and apoptosis-related p... Cancer
T1812 KX1-004 KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective dru... Cancer
T1803 GNF-5 GNF-5, an analogue of GNF-2 with improved pharmacokinetic properties, is a selective ... Other
T1606 Fasudil Fasudil hydrochloride (INN) is a potent Rho-kinase inhibitor and vasodilator. Since i... Nervous system
T1527 Gliclazide Gliclazide is a whole-cell beta-cell ATP-sensitive potassium currents blocker with an... Metabolism system
T1448L Dasatinib monohydrate Dasatinib is an oral dual BCR/ABL and Src family tyrosine kinase inhibitor approved f... Cancer
T0979 Dequalinium chloride Dequalinium Chloride is a selective blocker of apamin-sensitive K+ channels. Respiratory system
T6348 NVP-BHG712 NVP-BHG712 is a specific EphB4 inhibitor with ED50 of 25 nM that discriminates betwee... Cancer
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