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AG-1478  
Catalog No. T2047    CAS 153436-53-4
Pack Size
Availability
Price/USD
Quantity
5mg
In Stock
45.00
25mg
In Stock
132.00
50mg
In Stock
237.00
10mM * 1mL (in DMSO)
In Stock
47.00
10mg
In Stock
66.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet HNMR MSDS
Biological Activity:

Product Description:

AG-1478 (Tyrphostin AG-1478) is a selective EGFR inhibitor with IC50 of 3 nM in cell-free assays, almost no activity on HER2-Neu, PDGFR, Trk, Bcr-Abl and InsR.

Target:
PDGFR; HER2; EGFR;
Research Area:
Cancer
Chemical Information:
Molecular Weight 315.75
Formula C16H14ClN3O2
CAS Number 153436-53-4
Solubility Ethanol: 13 mg/mL (41.17 mM); DMSO: 25 mg/mL (79.17 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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