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Home > Chromatin/Epigenetic > EGFR > AG-490
AG-490  
Catalog No. T2600    CAS 133550-30-8
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Price/USD
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10mg
In stock
43.00
25mg
In stock
60.00
50mg
In stock
75.00
100mg
In stock
98.00
200mg
In stock
170.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
47.00
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Documents and Quality Management
Purity:98.60% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

AG-490 (Tyrphostin AG 490) is an inhibitor of EGFR with IC50 of 0.1 μM, 135-fold more selective for EGFR versus ErbB2, also inhibits JAK2 with no activity to Lck, Lyn, Btk, Syk and Src.

Target:
ErbB2; JAK2; EGFR;
Research Area:
Other
Chemical Information:
Molecular Weight 294.3
Formula C17H14N2O3
CAS Number 133550-30-8
Solubility DMSO: 58mg/ml(197.08 mM);Water: <1mg/ml;Ethanol: 6mg/ml(20.39 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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