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AT9283  
Catalog No. T3068    CAS 896466-04-9
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2mg
In stock
51.00
5mg
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77.00
10mg
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136.00
25mg
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232.00
50mg
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408.00
100mg
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689.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
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65.00
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Documents and Quality Management
Purity:98.45% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

AT9283 is a potent JAK2/3 inhibitor with IC50 of 1.2 nM/1.1 nM in cell-free assays; also potent to Aurora A/B, Abl(T315I). Phase 2.

Target:
VEGFR3/FLT4; FGFR2; GSK-3β; Abl1; Aurora B; Aurora A; JAK2; JAK3;
Research Area:
Cancer
Chemical Information:
Molecular Weight 381.43
Formula C19H23N7O2
CAS Number 896466-04-9
Solubility DMSO: 76mg/ml(199.25 mM);Water: <1mg/ml;Ethanol: 38mg/ml(99.63 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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