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Axitinib  
Catalog No. T1452    CAS 319460-85-0
Pack Size
Availability
Price/USD
Quantity
50mg
In Stock
78.00
100mg
In Stock
144.00
10mM * 1mL (in DMSO)
In Stock
53.00
10mg
In Stock
34.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.61% COA Datasheet HNMR HPLC LCMS
Biological Activity:

Product Description:

Axitinib is an oral, potent, and selective inhibitor of vascular endothelial growth factor receptors (VEGFR) 1, 2, and 3. Axitinib is marketed under the name Inlyta?, and if one previous systemic therapy for kidney cell cancer has failed, axitinib is indicated.

Target:
VEGFR3; VEGFR2; VEGFR1; PDGFRβ; c-Kit;
Research Area:
Cancer
Chemical Information:
Molecular Weight 386.47
Formula C22H18N4OS
CAS Number 319460-85-0
Solubility DMSO: 35mg/ml(90.56 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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