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Home > Tyrosine Kinase/Adaptors > PDGFR > CP-673451
CP-673451  
Catalog No. T6091    CAS 343787-29-1
Pack Size
Availability
Price/USD
Quantity
2mg
In Stock
71.00
10mg
In Stock
194.00
25mg
In Stock
376.00
50mg
In Stock
665.00
10mM * 1mL (in DMSO)
In Stock
94.00
5mg
In Stock
115.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.88% COA Datasheet HNMR HPLC
Biological Activity:

Product Description:

CP-673451 is a selective inhibitor of PDGFRα/β with IC50 of 10 nM/1 nM, exhibits >450-fold selectivity over other angiogenic receptors, has antiangiogenic and antitumor activity.

Target:
VEGFR2; VEGFR1; PDGFRβ; PDGFRα; c-Kit;
Research Area:
Cancer
Chemical Information:
Molecular Weight 417.50
Formula C24H27N5O2
CAS Number 343787-29-1
Solubility DMSO:28 mg/mL warmed (67.06 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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