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Home > Chromatin/Epigenetic > Pim > CX-6258 hydrochloride
CX-6258 hydrochloride  
Catalog No. T6148    CAS 1353859-00-3
Pack Size
Availability
Price/USD
Quantity
2mg
9 days
71.00
10mg
9 days
201.00
25mg
9 days
358.00
50mg
9 days
568.00
10mM * 1mL (in DMSO)
9 days
94.00
5mg
9 days
120.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

CX-6258 HCl is a potent, orally efficacious pan-Pim kinase inhibitor with IC50 of 5 nM, 25 nM and 16 nM for Pim1, Pim2, and Pim3, respectively.

Target:
Pim3; Pim2; Pim1;
Research Area:
Cancer
Chemical Information:
Molecular Weight 498.40
Formula C26H24ClN3O3·HCl
CAS Number 1353859-00-3
Solubility DMSO:57 mg/mL warmed (114.36 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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