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Home > Chromatin/Epigenetic > Pim > CX-6258
CX-6258  
Catalog No. T6148    CAS 1202916-90-2
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Availability
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5mg
9 days
102.00
10mg
9 days
136.00
25mg
9 days
221.00
50mg
9 days
383.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
9 days
112.00
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Documents and Quality Management
Purity:97.98% COA Datasheet HNMR
Biological Activity:

Product Description:

CX-6258 HCl is a potent, orally efficacious pan-Pim kinase inhibitor with IC50 of 5 nM, 25 nM and 16 nM for Pim1, Pim2, and Pim3, respectively.

Target:
Pim3; Pim2; Pim1;
Research Area:
cancer
Chemical Information:
Molecular Weight 498.4
Formula C26H24ClN3O3
CAS Number 1202916-90-2
Solubility DMSO: 57mg/ml(114.37 mM);Water: 89mg/ml(178.57 mM);Ethanol: 1mg/ml(2.01 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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