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Home > Chromatin/Epigenetic > Pim > CX-6258
CX-6258  
Catalog No. T1834    CAS 1202916-90-2
Pack Size
Availability
Price/USD
Quantity
10mg
9 days
142.00
50mg
9 days
441.00
10mM * 1mL (in DMSO)
9 days
99.00
25mg
9 days
240.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet HNMR
Biological Activity:

Product Description:

CX-6258 is a potent, orally efficacious Pim 1/2/3 kinase(IC50=5 nM/25 nM/16 nM) inhibitor with excellent biochemical potency and kinase selectivity

Target:
Pim3; Pim2; Pim1;
Research Area:
Other
Chemical Information:
Molecular Weight 461.94
Formula C26H24ClN3O3
CAS Number 1202916-90-2
Solubility DMSO > 10 mM
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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