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Home > Chromatin/Epigenetic > JAK > Cerdulatinib hydrochloride
Cerdulatinib hydrochloride  
Catalog No. T6104    CAS 1369761-01-2
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2mg
9 days
45.00
5mg
9 days
80.00
10mg
9 days
120.00
25mg
9 days
205.00
50mg
9 days
360.00
200mg
9 days
800.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
9 days
163.00
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Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

Cerdulatinib (PRT-062070) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of 12 nM/6 nM/8 nM/0.5 nM and 32 nM for JAK1/JAK2/JAK3/TYK2 and Syk, respectively. Also inhibits 19 other tested kinases with IC50 less than 200 nM.

Target:
TYK2; MST1; MLK1; Fms; ARK5;
Research Area:
Cancer
Chemical Information:
Molecular Weight 482
Formula C20H28ClN7O3S
CAS Number 1369761-01-2
Solubility DMSO: 43mg/ml(89.21 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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