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Home > Chromatin/Epigenetic > JAK > Decernotinib(VX-509)
Decernotinib(VX-509)  
Catalog No. T2636    CAS 944842-54-0
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2mg
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51.00
5mg
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77.00
10mg
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128.00
25mg
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230.00
50mg
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425.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
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66.00
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Documents and Quality Management
Purity:99.50% COA Datasheet HNMR HPLC
Biological Activity:

Product Description:

Decernotinib(VX-509; VRT-831509) is a potent and selective Janus kinase 3 (JAK3) inhibitor with Ki of 2.5 nM; IC50 is 50-170 nM in cellular assays.

Target:
JAK3;
Research Area:
Cancer
Chemical Information:
Molecular Weight 392.38
Formula C18H19F3N6O
CAS Number 944842-54-0
Solubility DMSO: 78mg/ml(198.79 mM);Water: <1mg/ml;Ethanol: 20mg/ml(50.97 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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