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Home > Chromatin/Epigenetic > JAK > GLPG0634 analogue
GLPG0634 analogue  
Catalog No. T3076    CAS 1206101-20-3
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1mg
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68.00
2mg
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102.00
5mg
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170.00
10mg
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298.00
25mg
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522.00
50mg
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935.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
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154.00
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Documents and Quality Management
Purity:99.50% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

GLPG0634 analogue is a selective JAK1 inhibitor with IC50 of 10 nM, 28 nM, 810 nM, and 116 nM for JAK1, JAK2, JAK3, and TYK2, respectively. Phase 2.

Target:
JAK3; JAK2; JAK1;
Research Area:
Cancer
Chemical Information:
Molecular Weight 425.5
Formula C21H23N5O3S
CAS Number 1206101-20-3
Solubility DMSO: 0.1mg/ml(0.24 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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