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Home > JAK/STAT signaling > c/Kit > KI8751
KI8751  
Catalog No. T2446    CAS 228559-41-9
Pack Size
Availability
Price/USD
Quantity
10mg
In Stock
74.00
50mg
In Stock
218.00
10mM * 1mL (in DMSO)
In Stock
69.00
25mg
In Stock
128.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.90% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

Ki8751 is a potent and selective inhibitor of VEGFR2 with IC50 of 0.9 nM, >40-fold selective for VEGFR2 than c-Kit, PDGFRα and FGFR-2, little activity to EGFR, HGFR and InsR.

Target:
VEGFR2; HGFR; EGFR ; FGFR2; PDGFRα ; c-Kit;
Research Area:
Cancer
Chemical Information:
Molecular Weight 469.41
Formula C24H18F3N3O4
CAS Number 228559-41-9
Solubility DMSO: 47mg/ml(100.13 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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