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Home > Chromatin/Epigenetic > FLT3 > Gandotinib (LY2784544)
Gandotinib (LY2784544)  
Catalog No. T2638    CAS 1229236-86-5
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Quantity
2mg
In stock
49.00
5mg
In stock
94.00
10mg
In stock
162.00
25mg
In stock
284.00
50mg
In stock
502.00
100mg
In stock
850.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
103.00
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Documents and Quality Management
Purity:99.79% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

LY2784544(gandotinib) is a potent JAK2 inhibitor with IC50 of 3 nM, effective in JAK2V617F(Ki=0.245 nM), 8- and 20-fold selective versus JAK1 and JAK3.

Target:
JAK2(V617F); JAK3; TYK2; FGFR2; FLT4; JAK1; JAK2; FLT3;
Research Area:
Cancer
Chemical Information:
Molecular Weight 469.94
Formula C23H25ClFN7O
CAS Number 1229236-86-5
Solubility DMSO: 94mg/ml(200.03 mM);Water: <1mg/ml;Ethanol: 9mg/ml(19.15 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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