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Home > Tyrosine Kinase/Adaptors > c/Kit > Masitinib
Masitinib  
Catalog No. T2609    CAS 790299-79-5
Pack Size
Availability
Price/USD
Quantity
2mg
In Stock
27.00
10mg
In Stock
45.00
50mg
In Stock
99.00
100mg
In Stock
156.00
10mM * 1mL (in DMSO)
In Stock
48.00
5mg
In Stock
38.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.50% COA Datasheet HNMR HPLC LCMS MSDS
Biological Activity:

Product Description:

Masitinib is a novel inhibitor for Kit and PDGFRα/β with IC50 of 200 nM and 540 nM/800 nM, weak inhibition to ABL and c-Fms. Phase 3.

Target:
PDGFRβ; PDGFRα; Lyn B; Kit;
Research Area:
Cancer
Chemical Information:
Molecular Weight 498.64
Formula C28H30N6OS
CAS Number 790299-79-5
Solubility Ethanol: 4 mg/mL (8.02 mM); DMSO: 100 mg/mL (200.54 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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