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Mocetinostat  
Catalog No. T2512    CAS 726169-73-9
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5mg
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28.00
10mg
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43.00
25mg
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66.00
50mg
In stock
84.00
100mg
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135.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
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47.00
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Documents and Quality Management
Purity:99.74% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

Mocetinostat (MGCD0103) is a potent HDAC inhibitor with most potency for HDAC1 with IC50 of 0.15 μM in a cell-free assay, 2- to 10- fold selectivity against HDAC2, 3, and 11, and no activity to HDAC4, 5, 6, 7, and 8. Phase 2.

Target:
HDAC1 ; HDAC3; HDAC11; HDAC2;
Research Area:
Cancer
Chemical Information:
Molecular Weight 396.44
Formula C23H20N6O
CAS Number 726169-73-9
Solubility DMSO: 13mg/ml(32.79 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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