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Home > Stem Cells > JAK > Mubritinib (TAK 165)
Mubritinib (TAK 165)  
Catalog No. T6124    CAS 366017-09-6
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Availability
Price/USD
Quantity
10mg
In stock
43.00
25mg
In stock
75.00
50mg
In stock
145.00
100mg
In stock
272.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
47.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet HNMR
Biological Activity:

Product Description:

Mubritinib (TAK-165) is a potent inhibitor of HER2/ErbB2 with IC50 of 6 nM; no activity to EGFR, FGFR, PDGFR, JAK1, Src and Blk. Phase 1.

Target:
PDGFR; JAK1; HER2/ErbB2; FGFR; EGFR;
Research Area:
Cancer
Chemical Information:
Molecular Weight 468.47
Formula C25H23F3N4O2
CAS Number 366017-09-6
Solubility DMSO: 13mg/ml(27.75 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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