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Home > Tyrosine Kinase/Adaptors > c/Kit > OSI-930
OSI-930  
Catalog No. T2624    CAS 728033-96-3
Pack Size
Availability
Price/USD
Quantity
5mg
In Stock
86.00
25mg
In Stock
228.00
50mg
In Stock
339.00
10mM * 1mL (in DMSO)
In Stock
50.00
10mg
In Stock
156.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.77% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

OSI-930 is a potent inhibitor of Kit, KDR and CSF-1R with IC50 of 80 nM, 9 nM and 15 nM, respectively; also potent to Flt-1, c-Raf and Lck and low activity against PDGFRα/β, Flt-3 and Abl. Phase 1.

Target:
LCK; KDR; FLT1; CSF-1R; C-Raf;
Research Area:
Cancer
Chemical Information:
Molecular Weight 443.44
Formula C22H16F3N3O2S
CAS Number 728033-96-3
Solubility DMSO: 89mg/ml(200.7 mM);Water: <1mg/ml;Ethanol: 3mg/ml(6.77 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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