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PP121  
Catalog No. T2415    CAS 1092788-83-4
Pack Size
Availability
Price/USD
Quantity
10mg
In Stock
79.00
50mg
In Stock
304.00
100mg
In Stock
368.00
10mM * 1mL (in DMSO)
In Stock
83.00
25mg
In Stock
218.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.67% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

PP-121 is a multi-targeted inhibitor of PDGFR, Hck, mTOR, VEGFR2, Src and Abl with IC50 of 2 nM, 8 nM, 10 nM, 12 nM, 14 nM and 18 nM, also inhibits DNA-PK with IC50 of 60 nM.

Target:
DNA-PK; Abl; Src; VEGFR2; mTOR; Hck; DGFR;
Research Area:
Cancer
Chemical Information:
Molecular Weight 319.36
Formula C17H17N7
CAS Number 1092788-83-4
Solubility Ethanol: 2 mg/mL (6.26 mM); DMSO: 64 mg/mL (200.4 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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