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Home > Tyrosine Kinase/Adaptors > FLT3 > Pacritinib (SB1518)
Pacritinib (SB1518)  
Catalog No. T6020    CAS 937272-79-2
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Availability
Price/USD
Quantity
2mg
In stock
40.00
5mg
In stock
77.00
10mg
In stock
102.00
25mg
In stock
189.00
50mg
In stock
298.00
100mg
In stock
468.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
144.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

Pacritinib (SB1518) is a potent and selective inhibitor of Janus Kinase 2 (JAK2) and Fms-Like Tyrosine Kinase-3 (FLT3) with IC50s of 23 and 22 nM in cell-free assays, respectively. Phase 3.

Target:
JAK2; JAK2(V617F); FLT3; FLT3(D835Y);
Research Area:
Cancer
Chemical Information:
Molecular Weight 472.58
Formula C28H32N4O3
CAS Number 937272-79-2
Solubility DMSO: 11mg/ml(23.28 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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