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Quisinostat (JNJ-26481585)  
Catalog No. T6055    CAS 875320-29-9
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Price/USD
Quantity
2mg
In stock
54.00
5mg
In stock
102.00
10mg
In stock
179.00
25mg
In stock
268.00
50mg
In stock
357.00
100mg
In stock
527.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
112.00
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Documents and Quality Management
Purity:99.00% COA Datasheet HNMR
Biological Activity:

Product Description:

Quisinostat (JNJ-26481585) is a novel second-generation HDAC inhibitor with highest potency for HDAC1 with IC50 of 0.11 nM, modest potent to HDACs 2, 4, 10, and 11; greater than 30-fold selectivity against HDACs 3, 5, 8, and 9 and lowest potency to HDACs 6 and 7. Phase 2.

Target:
HDAC4; HDAC2; HDAC11; HDAC10; HDAC1;
Research Area:
Cancer
Chemical Information:
Molecular Weight 394.48
Formula C21H26N6O2
CAS Number 875320-29-9
Solubility DMSO: 79 mg/mL (200.26 Mm
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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