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Home > Chromatin/Epigenetic > Tyrosine-Kinase-Adaptors-Others > TAK901
TAK901  
Catalog No. T2709    CAS 934541-31-8
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5mg
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89.00
10mg
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157.00
25mg
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279.00
50mg
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493.00
100mg
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748.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
99.00
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Documents and Quality Management
Purity:98.18% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

TAK-901 is a novel inhibitor of Aurora A/B with IC50 of 21 nM/15 nM. It is not a potent inhibitor of cellular JAK2, c-Src or Abl. Phase 1.

Target:
FGR; CLK2; c-Src; JAK3; Aurora B; Aurora A;
Research Area:
Cancer
Chemical Information:
Molecular Weight 504.64
Formula C28H32N4O3S
CAS Number 934541-31-8
Solubility DMSO: 101mg/ml(200.14 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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