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Tandutinib  
Catalog No. T1667    CAS 387867-13-2
Pack Size
Availability
Price/USD
Quantity
2mg
In Stock
20.00
10mM * 1mL (in DMSO)
In Stock
37.00
5mg
In Stock
40.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:99.00% COA Datasheet HNMR
Biological Activity:

Product Description:

Tandutinib (MLN518, CT53518) is a potent FLT3 antagonist with IC50 of 0.22 μM, also inhibits PDGFR and c-Kit, 15 to 20-fold higher potency for FLT3 versus CSF-1R and >100-fold selectivity for the same target versus FGFR, EGFR and KDR.

Target:
PDGFRβ; KDR; FLT3; CSF-1R; c-Kit;
Research Area:
Cancer
Chemical Information:
Molecular Weight 562.7
Formula C31H42N6O4
CAS Number 387867-13-2
Solubility Ethanol: 6 mg/mL (10.66 mM); DMSO: 5 mg/mL (8.88 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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