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Home > Tyrosine Kinase/Adaptors > c/Kit > Amuvatinib(MP470)
Amuvatinib(MP470)  
Catalog No. T2516    CAS 850879-09-3
Pack Size
Availability
Price/USD
Quantity
2mg
In Stock
72.00
10mg
In Stock
192.00
50mg
In Stock
509.00
10mM * 1mL (in DMSO)
In Stock
95.00
5mg
In Stock
115.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet HNMR MSDS
Biological Activity:

Product Description:

Amuvatinib (MP-470) is a potent and multi-targeted inhibitor of c-Kit, PDGFRα and Flt3 with IC50 of 10 nM, 40 nM and 81 nM, respectively. Phase 2.

Target:
PDGFRα (V561D); FLT3 (D835Y); c-Kit (D816H);
Research Area:
Cancer
Chemical Information:
Molecular Weight 447.51
Formula C23H21N5O3S
CAS Number 850879-09-3
Solubility DMSO: 32 mg/mL (71.5 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

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Reference

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