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SB408124  
Catalog No. T6658    CAS 288150-92-5
Pack Size
Availability
Price/USD
Quantity
5mg
9 days
50.00
10mM * 1mL (in DMSO)
9 days
70.00
100mg
9 days
285.00
Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.

Target:
OX1 (whole cell); OX1 (membrane);
Research Area:
Nervous system
Chemical Information:
Molecular Weight 356.37
Formula C19H18F2N4O
CAS Number 288150-92-5
Solubility DMSO:36 mg/mL (101.01 mM)
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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