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Home > Chromatin/Epigenetic > RET > TG101209
TG101209  
Catalog No. T3065    CAS 936091-14-4
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2mg
In stock
31.00
5mg
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60.00
10mg
In stock
94.00
25mg
In stock
133.00
50mg
In stock
213.00
100mg
In stock
383.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
In stock
66.00
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Documents and Quality Management
Purity:99.50% COA Datasheet HNMR HPLC MSDS
Biological Activity:

Product Description:

TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM, less potent to Flt3 and RET with IC50 of 25 nM and 17 nM in cell-free assays, ~30-fold selective for JAK2 than JAK3, sensitive to JAK2V617F and MPLW515L/K mutations.

Target:
RET; JAK3; JAK2; FLT3;
Research Area:
Cancer
Chemical Information:
Molecular Weight 509.67
Formula C26H35N7O2S
CAS Number 936091-14-4
Solubility DMSO: 102mg/ml(200.13 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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