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Compound Libraries Bioactive Compound Library

Bioactive Compound Library

Catalog No. L4000
  Library Compound List   Excel SDF

It contains more than 7739 small molecule compounds, with known biological activities causing biological reaction in cells, tissue even whole body, including Clinical compound library (L3400), Preclinical compound library (L3410), and Approved drug library (L1000). All compounds have clear targets and detailed information description, which is the key point to drug research and development like drug repurposing, small molecule inducing stem cell differentiation, and target identification in mechanism interrogation.

Many scientists have identified small molecules that can regulate cell fate and function, and stem cell differentiation by screening annotated bioactive compound library with confirmed activity and known targets. Recent advances in iPSC technology have made reprogramming of somatic cells towards pluripotency possible and simpler. Using both phenotypic screening and hypothesis-driven approaches, a growing number of compounds have been identified that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules with success in cardiomyocyte differentiation and proliferation, neural progenitor cells, etc.

In the library, we provide the peptides and other drug molecules with low solution stability in the form of dry powder (set as Part B) in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 57926.00
250 μL * 10 mM (in DMSO) 96698.00
1 mg 96698.00
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Product Description

  • A collection of 7739 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
  • All compounds have clear targets;
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • Covers various disease research areas, such as Cancer, Metabolism, Immunology and Cardiovascular system, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
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Library Composition

AChR (179)
5-HT Receptor (158)
COX (133)
Adrenergic Receptor (132)
Antibiotic (119)
Antibacterial (115)
Endogenous Metabolite (100)
DNA/RNA Synthesis (99)
Dopamine Receptor (95)
PI3K (89)
EGFR (88)
VEGFR (86)
Histamine Receptor (81)
Estrogen/progestogen Receptor (75)
CDK (68)
Sodium Channel (67)
Potassium Channel (66)
Autophagy (64)
NF-κB (59)
P450 (57)
Calcium Channel (55)
HDAC (54)
Bcr-Abl (53)
GABA Receptor (52)
JAK (52)
PDGFR (51)
Dehydrogenase (51)
Src (51)
PPAR (50)
Glucocorticoid Receptor (49)
Antioxidant (49)
Topoisomerase (49)
mTOR (48)
PDE (47)
FLT (46)
FGFR (45)
Microtubule Associated (45)
TNF (45)
Epigenetic Reader Domain (43)
c-Kit (43)
Histone Methyltransferase (40)
HIV Protease (40)
GluR (39)
GR (39)
Vitamin (38)
p38 MAPK (37)
Raf (37)
ERK (36)
Akt (35)
RAAS (35)
ALK (33)
STAT (33)
Wnt/beta-catenin (32)
ATPase (32)
c-Met/HGFR (32)
ribosome (32)
PKC (31)
MAO (30)
Antifungal (30)
GSK-3 (30)
TRP/TRPV Channel (30)
Tyrosine Kinases (29)
Androgen Receptor (29)
MMP (28)
NMDAR (28)
Norepinephrine (26)
IL Receptor (26)
Opioid Receptor (25)
Aurora Kinase (25)
BCL (25)
Carbonic Anhydrase (25)
DNA-PK (25)
GPR (24)
Antifection (24)
HSP (24)
MEK (24)
ROS (23)
IκB/IKK (22)
HCV Protease (21)
HER (21)
Amino Acids and Derivatives (21)
AMPK (21)
DNA Alkylation (21)
Sirtuin (21)
TGF-beta/Smad (20)
Antiviral (20)
Prostaglandin Receptor (20)
PKA (19)
Phospholipase (19)
PARP (19)
JNK (19)
TAM Receptor (19)
Tyrosinase (19)
S6 Kinase (19)
HIF (18)
p53 (18)
ATM/ATR (18)
Caspase (18)
Glucokinase (18)
P2 Receptor (17)
ROCK (17)
Hedgehog/Smoothened (17)
IGF-1R (16)
MRP (16)
Reverse Transcriptase (16)
Gamma-secretase (16)
CaMK (16)
Apoptosis (16)
Serine Protease (16)
Trk receptor (16)
Transferase (15)
Syk (15)
BTK (15)
Cannabinoid Receptor (15)
Casein Kinase (15)
Cysteine Protease (15)
DUB (15)
Proteasome (15)
Mdm2 (15)
Histone Demethylase (15)
Lipoxygenase (14)
NOS (14)
c-RET (14)
CXCR (14)
Thrombin (14)
Retinoid Receptor (14)
Beta Amyloid (13)
Adenosine Receptor (13)
NADPH (13)
Phosphatase (13)
Reductase (12)
Parasite (12)
AhR (12)
Chk (12)
CCR (12)
DHFR (12)
FAK (12)
TLR (12)
Serine/threonin kinase (11)
S1P Receptor (11)
DPP-4 (11)
CFTR (11)
Apoptosis inducer (11)
LRRK2 (11)
MAPK (11)
Integrin (11)
HMG-CoA Reductase (10)
Proton pump (10)
PLK (10)
DNA gyrase (10)
Sigma receptor (10)
Thyroid hormone receptor(THR) (10)
SGLT (9)
DNA Methyltransferase (9)
Aromatase (9)
CAT (9)
Chloride channel (9)
P-gp (9)
OX Receptor (9)
NOD (9)
IDO (9)
HSV (8)
HIF/HIF Prolyl-Hydroxylase (8)
HBV (8)
LTR (8)
Lipase (8)
Kinesin (8)
PDK (8)
Pim (8)
Rho (8)
ABC (8)
FAAH (8)
Factor Xa (8)
FXR (7)
c-Fms (7)
CSF-1R (7)
BACE (7)
PERK (7)
Lipid (7)
UGT (7)
Vasopressin Receptor (6)
transporter (6)
Liver X Receptor (6)
GPCR19 (6)
Hydroxylase (6)
Influenza Virus (6)
Platelet aggregation (6)
p97 (6)
PAI-1 (6)
c-Myc (6)
Annexin A (6)
Endothelin Receptor (6)
Fatty Acid Synthase (6)
Ferroptosis (6)
Free radical scavengers (5)
GNRH Receptor (5)
Ephrin Receptor (5)
CRM1 (5)
Nrf2 (5)
NAMPT (5)
PKM (5)
ROR (5)
IAP (5)
MPO (5)
Tie-2 (5)
Telomerase (5)
SGK (4)
Monocarboxylate transporter (4)
MLK (4)
LPA Receptor (4)
LDL (4)
PYK2 (4)
Protease-activated Receptor (4)
Porcupine (4)
Neurokinin receptor (4)
OCT (4)
PAK (4)
DprE1 (4)
DYRK (4)
E1/E2/E3 Enzyme (4)
cholecystokinin (4)
cell cycle arrest (4)
Cell wall (4)
CETP (4)
BMI-1 (3)
cAMP (3)
Carboxypeptidase(CPG2) (3)
Arginase (3)
ACAT (3)
Acetyl-CoA Carboxylase (3)
ACK (3)
advanced glycation end products (3)
Aminopeptidase (3)
Dynamin (3)
Decarboxylase (3)
DNA (3)
GRK (3)
GST (3)
Glucagon Receptor (3)
GluCls (3)
PD-1/PD-L1 (3)
PAFR (3)
Na-K-Cl cotransporter (3)
Nucleoside Antimetabolite/Analog (3)
NPC1L1 (3)
PGE Synthase (3)
Phosphorylase (3)
Ras (3)
LIM Kinase (3)
Monoamine Transporter (3)
MNK (3)
MT Receptor (3)
MTH1 (3)
Mitophagy (3)
Hck (3)
Histone Acetyltransferase (2)
Immunology & Inflammation related (2)
Mitochondrial Metabolism (2)
Melatonin Receptor (2)
KSP (2)
lysosomal autophagy (2)
PED (2)
OAT (2)
NADPH-oxidase (2)
Gap Junction Protein (2)
GTPase (2)
Glutathione reductase (2)
GlyT (2)
Discoidin Domain Receptor (DDR) (2)
Acyltransferase (2)
ASK (2)
ATP Citrate Lyase (2)
Bombesin Receptor (2)
BCRP (2)
CaSR (2)
Survivin (2)
Transaminase (2)
VDA (2)
Wee1 (2)
Wnk (2)
Xanthine Oxidase (1)
TOPK (1)
Thioredoxin (1)
Stemness kinase (1)
Somatostatin (1)
Serotonin Transporter (1)
Salt-Inducible Kinase (1)
CGRP Receptor (1)
Beta-Secretase (1)
BVDV (1)
Anion Exchanger (1)
Apelin receptor (1)
Adiponectin receptor (1)
AChE (1)
DNA Alkylator/Crosslinker (1)
CPT (1)
Electron transport (1)
FABP (1)
gp120/CD4 (1)
Glutaminase (1)
GSNOR (1)
GPX (1)
GHSR (1)
Fas/FasL (1)
FOXO1 (1)
N-Acetylglucosaminyltransferase (1)
NKCC (1)
NOD-like Receptor (NLR) (1)
P2X Receptor (1)
RAR/RXR (1)
PTEN (1)
MALT (1)
Keap1-Nrf (1)
LHRH (1)
MELK (1)
Monoamine Oxidase (1)
Integrase (1)
Interleukin Related (1)
IP3 Receptor  (1)
IRAK (1)
Hydrogenase (1)
iGluR (1)
Histone Acetylation (1)
hCE (1)
Hippo pathway (1)