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Compound Libraries Clinical Compound Library

Clinical Compound Library

Catalog No. L3400
  Library Compound List   Excel SDF

Clinical compound library is a collection of 1487 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 17640.00
250 μL * 10 mM (in DMSO) 29010.00
1 mg 29010.00
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Product Description

  • A unique collection of 1487 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
  • Shipped with blue ice
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Library Composition

PI3K (41)
VEGFR (36)
CDK (35)
EGFR (35)
JAK (28)
FLT (26)
FGFR (22)
mTOR (22)
c-Met/HGFR (20)
PDGFR (20)
Bcr-Abl (18)
HDAC (18)
5-HT Receptor (17)
c-Kit (17)
Src (17)
Aurora Kinase (16)
Akt (15)
p38 MAPK (15)
Tyrosine Kinases (14)
DNA/RNA Synthesis (14)
HSP (14)
GSK-3 (13)
HER (12)
ALK (12)
DNA-PK (11)
COX (11)
Epigenetic Reader Domain (11)
Estrogen/progestogen Receptor (11)
NF-κB (11)
Microtubule Associated (11)
PKC (11)
Raf (11)
PARP (10)
GPR (10)
Androgen Receptor (10)
AChR (10)
Chk (9)
Histamine Receptor (9)
MEK (9)
PPAR (9)
Syk (9)
TAM Receptor (9)
PDE (8)
HCV Protease (8)
ERK (8)
Endogenous Metabolite (8)
Dehydrogenase (8)
BCL (8)
Beta Amyloid (8)
BTK (8)
ATPase (7)
Autophagy (7)
Antibacterial (7)
c-RET (7)
GluR (7)
Histone Methyltransferase (7)
HIF (7)
MMP (7)
IDO (7)
P450 (7)
Potassium Channel (7)
Trk receptor (7)
TRP/TRPV Channel (6)
TLR (6)
Mdm2 (6)
PDK (6)
Pim (6)
PKA (6)
Phospholipase (6)
IGF-1R (6)
IL Receptor (6)
HIV Protease (6)
Gamma-secretase (6)
FAK (6)
Cannabinoid Receptor (6)
Caspase (6)
CCR (6)
CXCR (6)
Cysteine Protease (6)
Dopamine Receptor (6)
Adenosine Receptor (6)
Antiviral (6)
Calcium Channel (5)
Adrenergic Receptor (5)
CSF-1R (5)
Casein Kinase (5)
c-Fms (5)
FAAH (5)
GABA Receptor (5)
IκB/IKK (5)
p53 (5)
TNF (5)
STAT (5)
Sirtuin (5)
Prostaglandin Receptor (5)
RAAS (5)
ROS (5)
Transferase (5)
S1P Receptor (4)
S6 Kinase (4)
Serine Protease (4)
ROCK (4)
Proteasome (4)
Sodium Channel (4)
Sigma receptor (4)
TGF-beta/Smad (4)
Opioid Receptor (4)
P2 Receptor (4)
PLK (4)
IAP (4)
NMDAR (4)
LPA Receptor (4)
Histone Demethylase (4)
DNA Alkylation (4)
Antibiotic (4)
AMPK (4)
ATM/ATR (4)
BACE (3)
CFTR (3)
cholecystokinin (3)
CRM1 (3)
CETP (3)
Carbonic Anhydrase (3)
HIF/HIF Prolyl-Hydroxylase (3)
Hedgehog/Smoothened (3)
DUB (3)
Glucocorticoid Receptor (3)
Glucokinase (3)
NADPH (3)
Lipoxygenase (3)
Liver X Receptor (3)
JNK (3)
Kinesin (3)
HSV (3)
Hydroxylase (3)
P-gp (3)
OX Receptor (3)
Tie-2 (3)
transporter (3)
Wnt/beta-catenin (3)
Vitamin (2)
UGT (2)
Vasopressin Receptor (2)
Topoisomerase (2)
SGLT (2)
PYK2 (2)
Ras (2)
Retinoid Receptor (2)
Reverse Transcriptase (2)
PAK (2)
Parasite (2)
NAMPT (2)
Norepinephrine (2)
NOS (2)
Phosphatase (2)
Integrin (2)
KSP (2)
LTR (2)
DprE1 (2)
FXR (2)
Endothelin Receptor (2)
Antioxidant (2)
ATP Citrate Lyase (1)
Apoptosis (1)
Apoptosis inducer (1)
ASK (1)
CaMK (1)
Bombesin Receptor (1)
Antifection (1)
Antifungal (1)
Amino Acids and Derivatives (1)
Aminopeptidase (1)
advanced glycation end products (1)
AhR (1)
Acyltransferase (1)
ACAT (1)
Acetyl-CoA Carboxylase (1)
Ephrin Receptor (1)
DPP-4 (1)
DNA Methyltransferase (1)
Discoidin Domain Receptor (DDR) (1)
cell cycle arrest (1)
CGRP Receptor (1)
GlyT (1)
GNRH Receptor (1)
DYRK (1)
Ferroptosis (1)
GR (1)
GSNOR (1)
HBV (1)
Hck (1)
lysosomal autophagy (1)
MAO (1)
MELK (1)
Mitophagy (1)
MLK (1)
NADPH-oxidase (1)
MNK (1)
Monocarboxylate transporter (1)
NOD (1)
NOD-like Receptor (NLR) (1)
LDL (1)
LHRH (1)
IRAK (1)
Influenza Virus (1)
PED (1)
PERK (1)
Porcupine (1)
Platelet aggregation (1)
Nrf2 (1)
OAT (1)
Neurokinin receptor (1)
p97 (1)
PAFR (1)
PAI-1 (1)
Rho (1)
SGK (1)
Reductase (1)
Proton pump (1)
Protease-activated Receptor (1)
Stemness kinase (1)
Survivin (1)
TOPK (1)
Thioredoxin (1)
Thrombin (1)
Thyroid hormone receptor(THR) (1)
VDA (1)
Wee1 (1)