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β-Amino Acid Imagabalin Hydrochloride

Catalog No. T16447 CAS 610300-00-0

Synonyms: PD-0332334

β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.

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β-Amino Acid Imagabalin Hydrochloride Chemical Structure

β-Amino Acid Imagabalin Hydrochloride, CAS 610300-00-0

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description	β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.
In vivo	β-Amino Acid Imagabalin Hydrochloride had been also in phase I clinical trials for the treatment of chronic kidney disease. β-Amino Acid Imagabalin Hydrochloride had been in phase III clinical trials for the treatment of generalized anxiety disorders.

Synonyms	PD-0332334
Molecular Weight	209.71
Formula	C9H20ClNO2
CAS No.	610300-00-0

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Birch M, et al. A Simplified Process for the Manufacture of Imagabalin Hydrochloride (PD-0332334), an α2δ-Ligand for the Treatment of Generalised Anxiety Disorder. Org. Process Res. Dev., 2011, 15 (6), pp 1358–1364

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

β-Amino Acid Imagabalin Hydrochloride 610300-00-0 Membrane transporter/Ion channel Metabolism Calcium Channel b-Amino Acid Imagabalin Hydrochloride β Amino Acid Imagabalin Hydrochloride PD0332334 βAmino Acid Imagabalin Hydrochloride beta-Amino Acid Imagabalin Hydrochloride PD 0332334 PD-0332334 inhibitor inhibit

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