Powder: -20°C for 3 years | In solvent: -80°C for 1 year
1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 39.00 | |
10 mg | In stock | $ 64.00 | |
25 mg | In stock | $ 107.00 | |
50 mg | In stock | $ 163.00 | |
100 mg | In stock | $ 278.00 | |
200 mg | In stock | $ 418.00 | |
500 mg | In stock | $ 682.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 44.00 |
Description | 1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM). |
Targets&IC50 | CYP1A1:0.18 μM, CYP1A2:0.32 μM, CYP2B1:0.04 μM |
In vitro | The Ki values of 1-Ethynylpyrene against P450 1A2, and 2B1 is 0.32 and 0.04 μM, respectively[1]. |
Molecular Weight | 226.27 |
Formula | C18H10 |
CAS No. | 34993-56-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 9.09 mg/mL (40.17 mM)
You can also refer to dose conversion for different animals. More
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1-Ethynylpyrene 34993-56-1 Metabolism P450 1A1 1 Ethynylpyrene 2B1 Inhibitor CYPs Cytochrome P450 1Ethynylpyrene inhibit 1A2 cytochromes inhibitor