Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AKR1C1-IN-1 is a human 20α-hydroxysteroid dehydrogenase (AKR1C1) inhibitor (Ki: 4 nM for AKR1C1).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 44.00 | |
2 mg | In stock | $ 64.00 | |
5 mg | In stock | $ 98.00 | |
10 mg | In stock | $ 163.00 | |
25 mg | In stock | $ 293.00 | |
50 mg | In stock | $ 478.00 | |
100 mg | In stock | $ 688.00 | |
500 mg | In stock | $ 1,420.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 116.00 |
Description | AKR1C1-IN-1 is a human 20α-hydroxysteroid dehydrogenase (AKR1C1) inhibitor (Ki: 4 nM for AKR1C1). |
Targets&IC50 | AKR1C4:18.2 μM (Ki), AKR1C1:4 nM (Ki), AKR1C3:4.2 μM (Ki), AKR1C2:87 nM (Ki) |
In vitro | AKR1C1-IN-1 inhibits the metabolism of progesterone that in AKR1C1-overexpressed BAECs (IC50:460 nM). |
Molecular Weight | 293.11 |
Formula | C13H9BrO3 |
CAS No. | 4906-68-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 27.5 mg/mL (93.82 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
AKR1C1-IN-1 4906-68-7 Metabolism NADPH inhibit AKR-1C1-IN-1 progesterone AKR1C1IN1 AKR1C1 IN 1 Inhibitor AKR1C1 inhibitor