Powder: -20°C for 3 years | In solvent: -80°C for 1 year
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 51.00 | |
2 mg | In stock | $ 74.00 | |
5 mg | In stock | $ 122.00 | |
10 mg | In stock | $ 198.00 | |
25 mg | In stock | $ 378.00 | |
50 mg | In stock | $ 557.00 | |
100 mg | In stock | $ 773.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 129.00 |
Description | APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively. |
Targets&IC50 | ratGPR119:33 nM (EC50), hGPR119:2.7 nM (EC50) |
Synonyms | APD 668 |
Molecular Weight | 477.51 |
Formula | C21H24FN5O5S |
CAS No. | 832714-46-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (94.24 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
APD668 832714-46-2 Endocrinology/Hormones GPCR/G Protein Membrane transporter/Ion channel Metabolism Potassium Channel GPR P450 Inhibitor CYPs diabetes Cytochrome P450 APD-668 GPR119 coupled G-protein steatohepatitis CYP2C9 G Protein-Coupled Receptor 119 APD 668 inhibit KcsA inhibitor