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AS2717638

Catalog No. T10381   CAS 2148339-28-8

AS2717638 is an orally active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50: 38 nM for hLPA5). It also significantly improves PGF2α-, PGE2-, and AMPA-induced allodynia.

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AS2717638 Chemical Structure
AS2717638, CAS 2148339-28-8
Pack Size Availability Price/USD Quantity
1 mg In stock $ 148.00
5 mg In stock $ 322.00
10 mg In stock $ 538.00
25 mg In stock $ 869.00
50 mg In stock $ 1,180.00
100 mg In stock $ 1,590.00
1 mL * 10 mM (in DMSO) In stock $ 353.00
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Purity: 98.67%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description AS2717638 is an orally active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50: 38 nM for hLPA5). It also significantly improves PGF2α-, PGE2-, and AMPA-induced allodynia.
Targets&IC50 hLPA5:38 nM
Molecular Weight 447.48
Formula C25H25N3O5
CAS No. 2148339-28-8

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 54mg/mL (120.7mM), sonification is recommended.

TargetMolReferences and Literature

1. Murai N, et al. Analgesic effects of novel lysophosphatidic acid receptor 5 antagonist AS2717638 in rodents. Neuropharmacology. 2017 Nov;126:97-107.

Related compound libraries

This product is contained In the following compound libraries:
Bioactive Compound Library Inhibitor Library Bioactive Compounds Library Max

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Keywords

AS2717638 2148339-28-8 Others AS-2717638 AS 2717638 inhibitor inhibit

 

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