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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10407 | Gartisertib | ATR inhibitor 2 | ATM/ATR |
ATR inhibitor 2 is an orally active, ATP-competitive, and selective ATR inhibitor (Ki <150 pM) with antitumor activity. ATR inhibitor 2 potently inhibits ATR-driven phosphorylated checkpoint kinase-1 (Chk1) phosphorylati... |