Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial agonist on ORL1 transfected in CHO cells, antagonizes the stimulation of [35S]-GTPgammaS binding to G proteins by noc/OFQ in membranes and sections of rat brain.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 295.00 | |
2 mg | In stock | $ 443.00 | |
5 mg | In stock | $ 667.00 | |
10 mg | In stock | $ 997.00 | |
25 mg | In stock | $ 1,480.00 | |
50 mg | In stock | $ 1,990.00 | |
100 mg | In stock | $ 2,690.00 |
Description | Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial agonist on ORL1 transfected in CHO cells, antagonizes the stimulation of [35S]-GTPgammaS binding to G proteins by noc/OFQ in membranes and sections of rat brain. |
In vivo | When administered intracerebroventricularly (i.c.v.), Ac-RYYRIK-NH inhibited spontaneous locomotor activity in mice with ID50 of 0.07 nmol, respectively[1]. |
Molecular Weight | 999.17 |
Formula | C46H74N14O11 |
CAS No. | TP1940L1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Ac-RYYRIK-NH2 acetate TP1940L1 Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor Ac-RYYRIK-NH2 Acetate Ac-RYYRIK-NH-2 acetate AcRYYRIKNH2 acetate Ac RYYRIK NH2 acetate inhibitor inhibit