Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 163.00 | |
5 mg | In stock | $ 347.00 | |
10 mg | In stock | $ 497.00 | |
25 mg | In stock | $ 793.00 | |
50 mg | In stock | $ 1,130.00 | |
100 mg | In stock | $ 1,520.00 | |
500 mg | In stock | $ 2,970.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 382.00 |
Description | Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction. |
Targets&IC50 | Ca2+ channel, N-type:14.23 μM (EC50), CDK2:3.34 μM (EC50) |
In vitro | Ca2+ channel agonist 1 (Compound 13d) exhibits a ca. 2-fold increased agonism and a 22-fold decreased cdk2 kinase activity versus the standard, (R)-roscovitine. |
Molecular Weight | 354.45 |
Formula | C19H26N6O |
CAS No. | 1402821-24-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 40 mg/mL (112.85 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Ca2+ channel agonist 1 1402821-24-2 Cell Cycle/Checkpoint Membrane transporter/Ion channel Metabolism Calcium Channel CDK Ca2+ channels Inhibitor inhibit Ca channels Cyclin dependent kinase Ca-2+ channel agonist 1 inhibitor