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CaMKP Inhibitor

Catalog No. T2159 CAS 52789-62-5

CaMKP Inhibitor can inhibit CaMKP.

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CaMKP Inhibitor, CAS 52789-62-5

Pack Size	Availability	Price/USD
1 mg	In stock	$ 48.00
2 mg	In stock	$ 58.00
5 mg	In stock	$ 79.00
10 mg	In stock	$ 137.00
25 mg	In stock	$ 254.00
50 mg	In stock	$ 371.00
100 mg	In stock	$ 512.00
1 mL * 10 mM (in DMSO)	In stock	$ 109.00

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Purity: 99.98%

Purity: 96.55%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

CaMKP Inhibitor can inhibit CaMKP.

Kinase Assay

Biacore study: Competition assay is performed on a Biacore S51. A Series S Sensor chip CM5 is utilized for the immobilization of a PentaHis antibody for capture of the His-tagged p53. The level of capture is ~200 response units (1 response unit corresponds to 1 pg of protein per mm 2). The concentration of MDM2 protein is kept constant at 300 nM. Nutlin-3 is dissolved in DMSO at 10 mM and further diluted to make a concentration series of Nutlin-3 in each MDM2 test sample. The assay is run at 25°C in running buffer (10 mM Hepes, 0.15 M NaCl, 2% DMSO). MDM2-p53 binding in the presence of Nutlin-3 is calculated as a percentage of binding in the absence of Nutlin-3 and IC50 is calculated

Molecular Weight	377.32
Formula	C10H12NNaO9S2
CAS No.	52789-62-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 34.48 mg/mL (101.04 mM), Sonification is recommended.

DMSO: 10 mM

References and Literature

1. Nishizawa, E., Wynalda, D., & Lednicer, D. (1973). NON-THROMBOGENIC SURFACE INHIBITING PLATELET ADHERENCE. ASAIO Journal, 19(1), 13-18. doi: 10.1097/00002480-197301900-00003

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Kinase Inhibitor Library Anti-Neurodegenerative Disease Compound Library Target-Focused Phenotypic Screening Library Bioactive Compounds Library Max NO PAINS Compound Library Neuronal Signaling Compound Library Bioactive Compound Library

Related Products

Related compounds with same targets

KN-92 phosphate Melatonin CaM kinase II inhibitor TFA salt Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base) W-5 hydrochloride KN-93 Phosphate Autocamtide 2 TFA(129198-88-5 free base) Trifluoperazine dihydrochloride

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Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

CaMKP Inhibitor 52789-62-5 Neuroscience CaMK inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.