Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ceefourin 1 is a highly selective multidrug resistance protein 4 (MRP4) inhibitor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 36.00 | |
2 mg | In stock | $ 51.00 | |
5 mg | In stock | $ 80.00 | |
10 mg | In stock | $ 122.00 | |
25 mg | In stock | $ 263.00 | |
50 mg | In stock | $ 409.00 | |
100 mg | In stock | $ 596.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 111.00 |
Description | Ceefourin 1 is a highly selective multidrug resistance protein 4 (MRP4) inhibitor. |
In vitro | Ceefourin 1 and Ceefourin 2, that inhibit transport of a broad range of MRP4 substrates, yet are highly selective for MRP4 over other ABC transporters, including P-glycoprotein (P-gp), ABCG2 (Breast Cancer Resistance Protein;?BCRP) and MRP1 (multidrug resistance protein 1;?ABCC1).?Both compounds are more potent MRP4 inhibitors in cellular assays than the most widely used inhibitor, MK-571, requiring lower concentrations to effect a comparable level of inhibition.?Furthermore, Ceefourin 1 and Ceefourin 2 have low cellular toxicity, and high microsomal and acid stability. |
Molecular Weight | 294.42 |
Formula | C11H10N4S3 |
CAS No. | 315702-40-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 11 mg/mL (37.36 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Ceefourin 1 315702-40-0 Immunology/Inflammation MRP P-glycoprotein chemosensitizers inhibit efflux protein resistance Ceefourin1 MRP4 HEK293 D-luciferin ABC ABCG2 P-gp multidrug MRP1 Inhibitor neuroblastoma Ceefourin-1 ABCC1 BCRP inhibitor