Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 39.00 | |
5 mg | In stock | $ 63.00 | |
10 mg | In stock | $ 107.00 | |
25 mg | In stock | $ 195.00 | |
50 mg | In stock | $ 370.00 | |
100 mg | In stock | $ 548.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 68.00 |
Description | Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM, respectively. |
Targets&IC50 | Ca2+ influx (AITC-evoked):14.3μM, Ca2+ influx (4-HNE-evoked):18.7 μM |
Synonyms | TCS 5861528 |
Molecular Weight | 369.42 |
Formula | C19H23N5O3 |
CAS No. | 332117-28-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mM
You can also refer to dose conversion for different animals. More
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