Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist. Deschloroclozapine binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 50.00 | |
10 mg | In stock | $ 80.00 | |
25 mg | In stock | $ 156.00 | |
50 mg | In stock | $ 289.00 | |
100 mg | In stock | $ 449.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 66.00 |
Description | Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist. Deschloroclozapine binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively. |
Targets&IC50 | M3Dq (human):6.3 nM(Ki), M4Di (human):4.2 nM(Ki) |
Molecular Weight | 292.38 |
Formula | C18H20N4 |
CAS No. | 1977-07-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (342.02 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Deschloroclozapine 1977-07-7 Neuroscience Serotonin Transporter inhibit Inhibitor Muscarinic acetylcholine receptor hM4Di hM3Dq muscarinic-based mAChR DREADDs inhibitor