Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Desmethyl Erlotinib (CP-473420) is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 48.00 | |
2 mg | In stock | $ 70.00 | |
5 mg | In stock | $ 117.00 | |
10 mg | In stock | $ 198.00 | |
25 mg | In stock | $ 349.00 | |
50 mg | In stock | $ 523.00 | |
100 mg | In stock | $ 757.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 129.00 |
Description | Desmethyl Erlotinib (CP-473420) is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM). |
Targets&IC50 | EGFR:2 nM |
Synonyms | OSI-420, CP-473420, O-Desmethyl Erlotinib |
Molecular Weight | 379.41 |
Formula | C21H21N3O4 |
CAS No. | 183321-86-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
H2O: < 1 mg/mL (insoluble or slightly soluble)
DMSO: 83 mg/mL (199.58 mM), warmed
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Desmethyl Erlotinib 183321-86-0 Angiogenesis JAK/STAT signaling Metabolism Tyrosine Kinase/Adaptors EGFR Drug Metabolite Inhibitor CP 373420 OSI-420 CP-373420 CP373420 inhibit CP473420 CP-473420 OSI420 O-Desmethyl Erlotinib CP 473420 OSI 420 inhibitor