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ENS-163 phosphate

Catalog No. T11204 CAS 117707-51-4

Synonyms: Sandoz ENS 163 phosphate, ENS 213-163, Thiopilocarpine phosphate

Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.

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ENS-163 phosphate, CAS 117707-51-4

Pack Size	Availability	Price/USD
25 mg	6-8 weeks	$ 1,520.00
50 mg	6-8 weeks	$ 1,980.00
100 mg	6-8 weeks	$ 2,500.00

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This compound is a customized synthesis product. We have a strong synthesis team with excellent synthesis technology and capabilities. However, due to various objective factors, there is a low probability that the synthesis will not be successful. If you need to learn more, please feel free to consult us, we will serve you wholeheartedly.

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.
In vivo	ENS-163, a selective muscarinic M1 agonist, enhances long-term potentiation (LTP) in rat hippocampal slices. This compound has been studied specifically for its effects on LTP in a rat hippocampal slice preparation.

Synonyms	Sandoz ENS 163 phosphate, ENS 213-163, Thiopilocarpine phosphate
Molecular Weight	322.32
Formula	C11H19N2O5PS
CAS No.	117707-51-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Boddeke EW, et al. SDZ ENS 163, a selective muscarinic M1 receptor agonist, facilitates the induction of long-term potentiation in rat hippocampal slices. Eur J Pharmacol. 1992 Nov 3;222(1):21-5.

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

ENS-163 phosphate 117707-51-4 Others Sandoz ENS-163 Phosphate Thiopilocarpine Phosphate ENS163 Phosphate Sandoz ENS163 Phosphate Sandoz ENS 163 phosphate ENS 213-163 ENS 163 Phosphate ENS-163 Phosphate Thiopilocarpine phosphate Sandoz ENS 163 Phosphate ENS163 phosphate ENS 163 phosphate inhibitor inhibit

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