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Ecabet Sodium

Catalog No. T2587 CAS 86408-72-2

Synonyms: TA-2711E, TA-2711

Ecabet Sodium (TA-2711) is a potential new agent in the management of distal colitis.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Ecabet Sodium, CAS 86408-72-2

Pack Size	Availability	Price/USD
10 mg	In stock	$ 43.00
25 mg	In stock	$ 68.00
50 mg	In stock	$ 97.00
100 mg	In stock	$ 143.00
200 mg	In stock	$ 209.00
500 mg	In stock	$ 358.00
1 mL * 10 mM (in DMSO)	In stock	$ 48.00

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Purity: 97.68%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Ecabet Sodium (TA-2711) is a potential new agent in the management of distal colitis.

Kinase Assay

The inhibition profile of Cabozantinib against a broad panel of 270 human kinases is determined using luciferase-coupled chemiluminescence, 33P-phosphoryl transfer, or AlphaScreen technology. Recombinant human full-length, glutathione S-transferase tag, or histidine tag fusion proteins are used, and IC50 values are determined by measuring phosphorylation of peptide substrate poly(Glu, Tyr) at ATP concentrations at or below the Km for each respective kinase. The mechanism of kinase inhibition is evaluated using the AlphaScreen Assay by determining the IC50 values over a range of ATP concentrations[2].

Synonyms	TA-2711E, TA-2711
Molecular Weight	402.48
Formula	C20H27NaO5S
CAS No.	86408-72-2

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 50 mg/mL (124.23 mM)

References and Literature

1. Lawrance IC. J Gastroenterol Hepatol. 2010 Jul;25(7):1182-4.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Clinical Compound Library Anti-Cancer Approved Drug Library Anti-Cancer Drug Library Anti-Neurodegenerative Disease Compound Library Drug Repurposing Compound Library Metabolism Compound Library Anti-Liver Cancer Compound Library FDA-Approved & Pharmacopeia Drug Library Cuproptosis Compound Library NF-κB Signaling Compound Library

Related Products

Related compounds with same targets

Cysteamine hydrochloride Lipoic acid Tofogliflozin (hydrate) Methylprednisolone Acetate Glabridin Anti-inflammatory agent 47 BNTA Sodium dichloroacetate

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Ecabet Sodium 86408-72-2 Immunology/Inflammation Metabolism Microbiology/Virology NF-Κb Reactive Oxygen Species Antibacterial Inhibitor TA-2711E inhibit TA-2711 TA2711 Ecabet Bacterial TA 2711 inhibitor

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