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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2280 | Endoxifen (Z-isomer) | Endoxifen Z-isomer | Potassium Channel , Estrogen/progestogen Receptor , Estrogen Receptor/ERR , EGFR , HER |
Endoxifen Z-isomer (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity. |