Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 60.00 | |
2 mg | In stock | $ 85.00 | |
5 mg | In stock | $ 128.00 | |
10 mg | In stock | $ 197.00 | |
25 mg | In stock | $ 332.00 | |
50 mg | In stock | $ 463.00 | |
100 mg | In stock | $ 683.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 143.00 |
Description | Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) . |
In vivo | Enzalutamide is an oral agent for the treatment of metastatic castration-resistant prostate cancer (mCRPC);?N-desmethyl enzalutamide is its active metabolite, which has clinically relevant anti-androgen capacities similar to enzalutamide, and carboxylic acid enzalutamide is an inactive metabolite. |
Molecular Weight | 451.39 |
Formula | C20H13F4N3O3S |
CAS No. | 1242137-15-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (55.38 mM)
You can also refer to dose conversion for different animals. More
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Enzalutamide carboxylic acid 1242137-15-0 Endocrinology/Hormones Metabolism Androgen Receptor Drug Metabolite prostate metastatic MDV3100 carboxylic acid cancer metabolite androgen Inhibitor receptor castration-resistant inhibit inhibitor