Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene. Fluorobexarotene is a potent retinoid-X-receptor (RXR) agonist, with a Ki value of 12 nM and an EC50 value of 43 nM for RXRα receptor. Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 183.00 | |
5 mg | In stock | $ 463.00 | |
10 mg | In stock | $ 683.00 | |
25 mg | In stock | $ 1,070.00 | |
50 mg | In stock | $ 1,450.00 | |
100 mg | In stock | $ 1,950.00 | |
500 mg | In stock | $ 3,890.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 373.00 |
Description | Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene. Fluorobexarotene is a potent retinoid-X-receptor (RXR) agonist, with a Ki value of 12 nM and an EC50 value of 43 nM for RXRα receptor. Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene. |
Targets&IC50 | RXRα:12 nM (Ki), RXRα:43 nM (EC50) |
Molecular Weight | 366.47 |
Formula | C24H27FO2 |
CAS No. | 1190848-23-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 32.4mg/mL (88.4mM), sonification/heating is recommended.
You can also refer to dose conversion for different animals. More
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Fluorobexarotene 1190848-23-7 Metabolism Retinoid Receptor inhibitor inhibit