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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5118 | Brilanestrant | GDC0810 , GDC 0810 , GDC-0810 , ARN-810 , RG 6046 | Estrogen/progestogen Receptor , Estrogen Receptor/ERR |
Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM). |